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BAY 73-1449
CAS No. 693790-96-4
BAY 73-1449 ( BAY73-1449; BAY 73-1449 )
产品货号. M27855 CAS No. 693790-96-4
BAY 73-1449 is a selective and potent antagonist of the prostacyclin receptor(IC50<0.1 nM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥2001 | 有现货 |
|
| 10MG | ￥3345 | 有现货 |
|
| 25MG | ￥5605 | 有现货 |
|
| 50MG | ￥7979 | 有现货 |
|
| 100MG | ￥10773 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称BAY 73-1449
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述BAY 73-1449 is a selective and potent antagonist of the prostacyclin receptor(IC50<0.1 nM).
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产品描述BAY 73-1449 is a selective and potent antagonist of the prostacyclin receptor(IC50<0.1 nM).(In Vivo):In male Wistar rats, BAY 73-1449 (0.1-1 mg/kg; i.v.) significantly reduced splenic shunt vessel outflow without affecting mesenteric inflow. BAY 73-1449 (1-5 mg/kg; s.c.) has no effects on portal pressures and the degree of porto-systemic shunting in rats.
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同义词BAY73-1449; BAY 73-1449
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通路Others
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靶点Other Targets
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受体RhoA; Lbc
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研究领域——
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适应症——
化学信息
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CAS Number693790-96-4
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分子量425.5
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分子式C26H23N3O3
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纯度>98% (HPLC)
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溶解度——
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SMILESOC(=O)[C@H](Cc1ccccc1)Nc1cc(ncn1)-c1ccc(OCc2ccccc2)cc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Francesca FANELLI, et al. Compounds and composition for use in the inhibition of the lbc-rhoa interaction, in particular for the treatment of cancer. WO2015028929A1.
产品手册
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